发明名称 PROCESS OF PRODUCING CYCLOALKYLCARBOXAMIDO-INDOLE COMPOUNDS
摘要 The present invention features processes for preparing compounds, such as ( R )-1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-N-(1-(2,3-dihydroxypropyl)-6-fluoro-2-(1-hydroxy-2-methylpropan-2-yl)-1H-indol-5-yl)cyclopropanecarboxamide (Compound 1), useful for treating CFTR mediated diseases such as cystic fibrosis.
申请公布号 EP2560954(A2) 申请公布日期 2013.02.27
申请号 EP20110729195 申请日期 2011.04.21
申请人 VERTEX PHARMACEUTICALS INCORPORATED 发明人 LEE, ELAINE, CHUNGMIN;TANOURY, GERALD, J.;HARRISON, CRISTIAN;LITTLER, BENJAMIN, JOSEPH;ROSE, PETER, JAMISON;HUGHES, ROBERT, MICHAEL;JUNG, YOUNG CHUN;SIESEL, DAVID, ANDREW;BELMONT, DANIEL, T.
分类号 C07D209/12;C07D317/60;C07D405/12 主分类号 C07D209/12
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