发明名称 Heterocyclidene acetamide derivative
摘要 A compound represented by formula (I′): (wherein m, n, and p each represent 0 to 2; q represents 0 or 1; R1 represents halogen, a hydrocarbon group, a heterocyclic group, an alkoxy group, an alkoxycarbonyl group, a sulfamoyl group, a CN group, an NO2 group, or the like; R2 represents halogen, amino, a hydrocarbon group, an aromatic heterocyclic group, or an oxo group; X1 represents O, —NR3—, or —S(O)r-; X2 represents a methylene group, O, —NR3—, or —S(O)r-; Q′ represents a heteroaryl group, a heteroarylalkyl group, a substituted aryl group, or an aralkyl group; Cycle moiety represents an aryl ring or a heteroaryl ring; and the wavy line represents an E-isomer or a Z-isomer), a salt of the compound, or a solvate of the compound or the salt. A pharmaceutical composition and a transient receptor potential type I (TRPV1) receptor antagonist each contain, as an active ingredient, at least one of the compound, a salt of the compound, and a solvate of the compound or the salt.
申请公布号 US8383839(B2) 申请公布日期 2013.02.26
申请号 US201113008456 申请日期 2011.01.18
申请人 MOCHIDA PHARMACEUTICAL CO., LTD.;UCHIDA HIDEHARU;KOSUGA NAOTO;SATOH TSUTOMU;HOTTA DAIDO;KAMINO TOMOYUKI;MAEDA YOSHITAKA;AMANO KEN-ICHI;AKADA YASUSHIGE 发明人 UCHIDA HIDEHARU;KOSUGA NAOTO;SATOH TSUTOMU;HOTTA DAIDO;KAMINO TOMOYUKI;MAEDA YOSHITAKA;AMANO KEN-ICHI;AKADA YASUSHIGE
分类号 C07D313/00;C07D309/00 主分类号 C07D313/00
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