发明名称 NOVEL UREA DERIVATIVES AS TEC KINASE INHIBITORS AND USES THEREOF
摘要 <p>Provided are urea compounds of formula (I) as Tec kinase inhibitors, in particular ITK (interleukin-2 inducible tyrosine kinase) inhibitors. Also provided herein are processes for preparing compounds described herein, intermediates used in their synthesis, pharmaceutical compositions thereof, and methods for treating or preventing diseases, conditions and/or disorders mediated by ITK.</p>
申请公布号 WO2013024427(A1) 申请公布日期 2013.02.21
申请号 WO2012IB54126 申请日期 2012.08.14
申请人 GLENMARK PHARMACEUTICALS S.A.;CHAUDHARI, SACHIN SUNDARLAL;THOMAS, ABRAHAM;ADIK, BHARAT GANGADHAR;DHONE, SACHIN VASANTRAO;WADEKAR, PRASHANT DILIP;KHAIRATKAR-JOSHI, NEELIMA;SHAH, DAISY MANISH 发明人 CHAUDHARI, SACHIN SUNDARLAL;THOMAS, ABRAHAM;ADIK, BHARAT GANGADHAR;DHONE, SACHIN VASANTRAO;WADEKAR, PRASHANT DILIP;KHAIRATKAR-JOSHI, NEELIMA;SHAH, DAISY MANISH
分类号 C07D403/12;A61K31/4184;A61P11/06;A61P37/08;C07D403/14 主分类号 C07D403/12
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