发明名称 TRICYCLIC PYRIDYL-VINYL-PYROLES AS PAR1 INHIBITORS
摘要 This disclosure relates to compounds of formula I: wherein R1, R2, R3, R4, X and Y have the meanings denoted in the disclosure. The compounds of formula I have antithrombotic activity and in particular inhibit the protease-activated receptor 1 (PAR1). The disclosure further relates to a method for producing the compound of formula I and to the use thereof as a pharmaceutical product.
申请公布号 EP2558465(A1) 申请公布日期 2013.02.20
申请号 EP20110715496 申请日期 2011.04.14
申请人 SANOFI 发明人 SCHOENAFINGER, KARL;STEINHAGEN, HENNING;SCHEIPER, BODO;HEINELT, UWE;WEHNER, VOLKMAR;HERRMANN, MATTHIAS
分类号 C07D471/14;A61K31/407;A61K31/437;A61K31/4985;A61K31/5383;A61P7/02;C07D487/14;C07D498/14 主分类号 C07D471/14
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