发明名称 |
ACID ADDITION SALTS OF THE 2-[2-[[(4-METHOXY-2,6-DIMETHYLPHENYL)S ULFONYL]-(METHYL)AMINO]ETHOXY]-N-METHYL-N-[3-(4-METHYLPIPERAZIN- 1-YL)CYCLOHEXYL] ACETAMIDE AND THE USE THEREOF AS BRADYKININ B1 RECEPTOR ANTAGONISTS. |
摘要 |
<p>The invention relates to the novel acid addition salts AB of the following free base of formula (A) or the enantiomer thereof with a physiologically acceptable acid B selected from the group consisting of hydrochloric acid, fumaric acid, and tartaric acid and to the polymorphs, hydrates, and solvates thereof.</p> |
申请公布号 |
MX2013000978(A) |
申请公布日期 |
2013.02.15 |
申请号 |
MX20130000978 |
申请日期 |
2011.08.04 |
申请人 |
BOEHRINGER INGELHEIM INTERNATIONAL GMBH.* |
发明人 |
JUERGEN SCHNAUBELT;WALDERMAR PFRENGLE;THORSTEN PACHUR;ULRIKE WERTHMANN;MANFRED BIRK |
分类号 |
C07D295/135;A61K31/495;A61P29/00 |
主分类号 |
C07D295/135 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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