ANHYDROUS AND HEMIHYDRATE CRYSTALLINE FORMS OF AN (R)-BACLOFEN PRODRUG, METHODS OF SYNTHESIS AND METHODS OF USE
摘要
<p>Crystalline (3R)-4-{[(1S)-2-methyl-1-(2-methylpropanoyloxy)propoxy]carbonylamino}-3-(4-chlorophenyl)butanoic acid anhydrate and crystalline (3R)-4-{[(1S)-2-methyl-1-(2-methylpropanoyloxy)propoxy]carbonylamino}-3-(4-chlorophenyl)butanoic acid hemihydrate, pharmaceutical compositions comprising such compounds, methods of making and methods of using the same are disclosed.</p>
申请公布号
WO2013023155(A1)
申请公布日期
2013.02.14
申请号
WO2012US50379
申请日期
2012.08.10
申请人
XENOPORT, INC.;RAILLARD, STEPHEN P;MANTHATI, SURESH K;JOSHI, SUDHIR
发明人
RAILLARD, STEPHEN P;MANTHATI, SURESH K;JOSHI, SUDHIR