发明名称 |
SOLID FORMS OF 3-(6-(1-(2,2-DIFLUOROBENZO[D][1,3]DIOXOL-5-YL) CYCLOPROPANECARBOXAMIDO)-3-METHYLPYRIDIN-2-YL)BENZOIC ACID |
摘要 |
<p>The present invention relates to a substantially a solid form of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid (Compound 1, Solvate Form A and Compound 1, HCl Salt Form A), processes for making such forms, pharmaceutical compositions thereof, and methods of treatment therewith.</p> |
申请公布号 |
EP2555754(A2) |
申请公布日期 |
2013.02.13 |
申请号 |
EP20110714625 |
申请日期 |
2011.04.07 |
申请人 |
VERTEX PHARMACEUTICALS INCORPORATED |
发明人 |
KESHAVARZ-SHOKRI, ALI;ZHANG, BEILI;KRAWIEC, MARIUSZ |
分类号 |
A61K9/16;A61K9/20;A61K9/28;C07D213/75;C07D405/12;C07D405/14 |
主分类号 |
A61K9/16 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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