发明名称 Salts of methyl 2-((R)-(3-chlorophenyl)((R)-1-((S)-2-(methylamino)-3-((R)-tetrahydro-2H-pyran-3-yl)propylcarbamoyl)piperidin-3-yl)methoxy)ethylcarbamate
摘要 Mucic acid salts of a compound represented by the following structural formula: are disclosed. In particular, single crystalline mucic acid salts of the compound represented by structural formula (I) are characterized by a variety of properties and physical measurements. Methods of producing the mucic acid salts, using the salts to antagonize one or more aspartic proteases, and methods of treating a number of aspartic protease mediated disorders using the salts are described herein.
申请公布号 US8372978(B2) 申请公布日期 2013.02.12
申请号 US20100851267 申请日期 2010.08.05
申请人 VITAE PHARMACEUTICALS, INC.;CLAREMON DAVID A.;SIMPSON ROBERT D.;JIA LANQI 发明人 CLAREMON DAVID A.;SIMPSON ROBERT D.;JIA LANQI
分类号 A61K31/453;A61P9/00;C07D413/12 主分类号 A61K31/453
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