| 发明名称 |
PREPARATION OF 13-CYCLOHEXYL-3-METHOXY-6-[METHYL-(2-{2-[METHYL-(S ULPHAMOYL)-AMINO]-ETHOXY}-ETHYL)-CARBAMOYL]-7<i>H</i>-INDOLO-[2, 1-a]-[2]-BENZAZEPINE-10-CARBOXYLIC ACID. |
| 摘要 |
<p>The present invention relates to an improved method for the preparation of 3-cyclohexyl-3-methoxy-6-[methyl-(2-{2-[methyl-(sulphamoyl)-ami no]-ethoxy}- ethyl)-carbamoyl]-7<i>H</i>-indolo-[2,1-a]-[2]-benzazepine-10-c arboxylic acid. The present invention also relates to a new compound, namely tert-butyl (methyl-{2-[2-(methylamino)-ethoxy]-ethyl}-sulphamoyl)-carbamat e, used in this improved method.</p> |
| 申请公布号 |
MX2012015198(A) |
申请公布日期 |
2013.02.11 |
| 申请号 |
MX20120015198 |
申请日期 |
2011.06.24 |
| 申请人 |
JANSSEN R&D IRELAND.* |
发明人 |
BONGARTZ, JEAN-PIERRE ANDRE MARC;NIESTE, PATRICK HUBERT J.;GOVAERTS, TOM CORNELIS HORTENSE |
| 分类号 |
C07D223/14 |
主分类号 |
C07D223/14 |
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