发明名称 AMIDINE COMPOUND OR SALT THEREOF
摘要 <p>The purpose of the present invention is to provide a novel compound which has an anti-fungal activity on pathogenic fungi including fungi belonging to the genus Candida, the genus Aspergillus and the genus Trichophyton and is useful as a medicinal agent. A compound represented by formula (I) (wherein A1 represents a nitrogen atom or a group represented by formula CR6; A2 and A3 are the same as or different from each other and independently represent a nitrogen atom or a group represented by formula CH; R1 represents an aryl group which may be substituted by 1 to 5 substituents independently selected from a substituent group (2) or the like; R2 and R3 are the same as or different from each other and independently represent a hydrogen atom, a halogen atom, a C1-6 alkyl group, a C1-6 haloalkyl group or a C1-6 alkoxy group; and R4 and R5 are the same as or different from each other and independently represent a hydrogen atom, a C1-6 haloalkyl group, a C1-6 alkyl group or the like) or a salt thereof is useful as an anti-fungal agent.</p>
申请公布号 WO2013018735(A1) 申请公布日期 2013.02.07
申请号 WO2012JP69249 申请日期 2012.07.27
申请人 TAISHO PHARMACEUTICAL CO., LTD.;TOYAMA CHEMICAL CO., LTD.;TANIKAWA TETSUYA;USHIKI YASUNOBU;USHIYAMA FUMIHITO;YAMAGUCHI TORU;ONO NAOYA;YAMAMOTO KEIKO;TSURUTA RISA;TSUTSUI YASUHIRO;FUJINO NORITOMO;MORI AYUMU 发明人 TANIKAWA TETSUYA;USHIKI YASUNOBU;USHIYAMA FUMIHITO;YAMAGUCHI TORU;ONO NAOYA;YAMAMOTO KEIKO;TSURUTA RISA;TSUTSUI YASUHIRO;FUJINO NORITOMO;MORI AYUMU
分类号 C07D277/28;A61K31/426;A61K31/427;A61K31/433;A61K31/4439;A61K31/454;A61K31/496;A61K31/497;A61K31/501;A61K31/506;A61K31/5377;A61P17/00;A61P31/10;C07D277/20;C07D277/30;C07D277/34;C07D277/48;C07D277/56;C07D285/08;C07D417/04;C07D417/06;C07D417/12 主分类号 C07D277/28
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