发明名称 |
C-17 AND C-3 MODIFIED TRITERPENOIDS WITH HIV MATURATION INHIBITORY ACTIVITY |
摘要 |
Compounds having drug and bio-affecting properties, their pharmaceutical compositions and methods of use are set forth. In particular, C-17 and C-3 modified triterpenoids that possess unique antiviral activity are provided as HIV maturation inhibitors, as represented by compounds of Formulas I, II and III: These compounds are useful for the treatment of HIV and AIDS.
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申请公布号 |
US2013035318(A1) |
申请公布日期 |
2013.02.07 |
申请号 |
US201213359727 |
申请日期 |
2012.01.27 |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY;REGUEIRO-REN ALICIA;LIU ZHENG;SWIDORSKI JACOB;SIN NY;VENABLES BRIAN LEE;SIT SING-YUEN;CHEN YAN;CHEN JIE;MEANWELL NICHOLAS A. |
发明人 |
REGUEIRO-REN ALICIA;LIU ZHENG;SWIDORSKI JACOB;SIN NY;VENABLES BRIAN LEE;SIT SING-YUEN;CHEN YAN;CHEN JIE;MEANWELL NICHOLAS A. |
分类号 |
C07J53/00;A61K31/565;A61K31/58;A61P31/18 |
主分类号 |
C07J53/00 |
代理机构 |
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地址 |
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