发明名称 C-17 AND C-3 MODIFIED TRITERPENOIDS WITH HIV MATURATION INHIBITORY ACTIVITY
摘要 Compounds having drug and bio-affecting properties, their pharmaceutical compositions and methods of use are set forth. In particular, C-17 and C-3 modified triterpenoids that possess unique antiviral activity are provided as HIV maturation inhibitors, as represented by compounds of Formulas I, II and III: These compounds are useful for the treatment of HIV and AIDS.
申请公布号 US2013035318(A1) 申请公布日期 2013.02.07
申请号 US201213359727 申请日期 2012.01.27
申请人 BRISTOL-MYERS SQUIBB COMPANY;REGUEIRO-REN ALICIA;LIU ZHENG;SWIDORSKI JACOB;SIN NY;VENABLES BRIAN LEE;SIT SING-YUEN;CHEN YAN;CHEN JIE;MEANWELL NICHOLAS A. 发明人 REGUEIRO-REN ALICIA;LIU ZHENG;SWIDORSKI JACOB;SIN NY;VENABLES BRIAN LEE;SIT SING-YUEN;CHEN YAN;CHEN JIE;MEANWELL NICHOLAS A.
分类号 C07J53/00;A61K31/565;A61K31/58;A61P31/18 主分类号 C07J53/00
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