MULTICOMPONENT CRYSTALLINE SYSTEM OF EZETIMIBE AND PROLINE
摘要
<p>Provided is a crystalline composition comprising a mixture of a compound of formula 1 (Ezetimibe) and proline or proline derivatives, or a hydrate/solvate thereof, as well as a process for obtaining the same. And a process for the purification of Ezetimibe is also disclosed.</p>
申请公布号
WO2013014604(A1)
申请公布日期
2013.01.31
申请号
WO2012IB53751
申请日期
2012.07.24
申请人
BASF SE;HAFNER, ANDREAS;HINTERMANN, TOBIAS;SZELAGIEWICZ, MARTIN;SIEBENHAAR, BERND;BLATTER, FRITZ;BASF (CHINA) COMPANY LIMITED
发明人
HAFNER, ANDREAS;HINTERMANN, TOBIAS;SZELAGIEWICZ, MARTIN;SIEBENHAAR, BERND;BLATTER, FRITZ