发明名称 |
SUBSTITUTED 4-{3-[6-AMINO-9-(3,4-DIHYDROXY-TETRAHYDRO-FURAN-2-YL)-9H-PURIN-2-YL]-PROP-2-YNYL}-PIPERIDINE-1-CARBOXYLIC ACID ESTERS AS A2AR AGONISTS |
摘要 |
<p>The present invention provides substituted 4-f 3-16-amino-9-(3,4-dihydroxy tetrahydro-furan-2-y1)-9H-purin-2-y11-prop-2-ynyl I -piperidine-l-carboxylic acid esters and pharmaceutical compositions containg the same that are selective agonists of A2A adenosine receptors (ARs). These compounds and compositions are useful as pharmaceutical agents.No Figure</p> |
申请公布号 |
SG186676(A1) |
申请公布日期 |
2013.01.30 |
申请号 |
SG20120093936 |
申请日期 |
2008.12.20 |
申请人 |
TROVIS PHARMACEUTICALS LLC |
发明人 |
THOMPSON, ROBERT;BEAUGLEHOLE, ANTHONY;SCHMIDTMANN, FRANK;RIEGER, JAYSON |
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