发明名称 Macrocyclic compound
摘要 The present invention provides a novel class of compounds that have the activity of inhibiting HSP90 enzyme and are useful as anti-cancer agents or such, and compounds that are useful as synthetic intermediates thereof. Specifically, the present invention provides compounds represented by the following formula (1), and pharmaceutically acceptable salts thereof: wherein X, R1, R2, R3, R4, R5, R6, R7, L1, L2, and L3 are as defined in the specification.
申请公布号 US8362236(B2) 申请公布日期 2013.01.29
申请号 US20080529222 申请日期 2008.02.29
申请人 CHUGAI SEIYAKU KABUSHIKI KAISHA;SHIMMA NOBUO;TSUKUDA TAKUO;KOYANO HIROSHI;SUDA ATSUSHI;HAYASE TADAKATSU;HADA KIHITO;KAWASAKI KEN-ICHI;KOMIYAMA SUSUMU;ONO NAOMI;YAMAZAKI TOSHIKAZU;SAITOH RYOICHI;KOHCHI MASAMI;HASEGAWA KIYOSHI 发明人 SHIMMA NOBUO;TSUKUDA TAKUO;KOYANO HIROSHI;SUDA ATSUSHI;HAYASE TADAKATSU;HADA KIHITO;KAWASAKI KEN-ICHI;KOMIYAMA SUSUMU;ONO NAOMI;YAMAZAKI TOSHIKAZU;SAITOH RYOICHI;KOHCHI MASAMI;HASEGAWA KIYOSHI
分类号 C07D497/08;A61K31/529;A61K31/53;A61K31/5377;A61P35/00;C07D513/08;C07D513/20 主分类号 C07D497/08
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