发明名称 DERIVATIVES OF 2-PYRIDIN-2-YL-PYRAZOL-3(2H)-ONE, PREPARATION AND THERAPEUTIC USE THEREOF
摘要 593797 Disclosed are substituted dihydropyrazolone derivatives of formula (I), wherein the substituents are as described within the specification. An examples of compounds of formula (I) is 2-[5-(piperidin-1-ylsulfonyl)pyridine-2-yl]-1,2,4,5,6,7-hexahydro-3H-indazol-3-one. Further disclosed is a process for preparing a compound of formula (I), a pharmaceutical composition comprising formula (I), and the use of a compound of formula (I) in the manufacture of a medicament for the treatment/prophylaxis of cardiovascular diseases, glaucoma, neurodegenerative diseases, etc.
申请公布号 NZ593797(A) 申请公布日期 2013.01.25
申请号 NZ20090593797 申请日期 2009.12.24
申请人 SANOFI 发明人 ALTENBURGER, JEAN-MICHEL;FOSSEY, VALERIE;ILLIANO, STEPHANE;MANETTE, GERALDINE
分类号 A61P27/06;A61K31/4162;C07D213/72;C07D213/77;C07D401/12;C07D403/04;C07D405/12;C07D409/12;C07D471/04;C07D491/04;C07D495/04;C07D513/04 主分类号 A61P27/06
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