发明名称 PROCESS FOR PREPARING ELETRIPTAN HYDROBROMIDE HAVING a-FORM
摘要 A process for preparation of eletriptan hydrobromide having a-form of formula (I) is described that includes reducing 3-((R)-1-methylpyrrolidin-2-yl)methyl)-5-((E)-2-(phenylsulfonyl)vinyl)-1H-indole of formula (II) in presence of a metal catalyst to the product of formula (III) and then converting to hydrobromide salt having a-form of formula (I).
申请公布号 US2013023672(A1) 申请公布日期 2013.01.24
申请号 US201013522850 申请日期 2010.03.31
申请人 VENTURI SRINIVASA RAO;KODALI HARI PRASAD;VENKATA SUBHRAMANIAN HARIHARAKRISHNAN;TADIMALLA VANKATA SRIHARI;POTLURI RAMESH BABU 发明人 VENTURI SRINIVASA RAO;KODALI HARI PRASAD;VENKATA SUBHRAMANIAN HARIHARAKRISHNAN;TADIMALLA VANKATA SRIHARI;POTLURI RAMESH BABU
分类号 C07D403/06 主分类号 C07D403/06
代理机构 代理人
主权项
地址
您可能感兴趣的专利