发明名称 |
SUBSTITUTED QUINAZOLINES, THE PREPARATION THEREOF AND THE USE THEREOF IN PHARMACEUTICAL COMPOSITIONS |
摘要 |
<p>The present invention relates to substituted quinazolines of formula (I) wherein X and Y are defined as in claim 1, the tautomers, stereoisomers, mixtures and salts thereof, which have valuable pharmacological properties, particularly an inhibitory effect on the activity of the enzyme dipeptidylpeptidase-IV (DPP-IV).</p> |
申请公布号 |
CA2841552(A1) |
申请公布日期 |
2013.01.24 |
申请号 |
CA20122841552 |
申请日期 |
2012.07.13 |
申请人 |
BOEHRINGER INGELHEIM INTERNATIONAL GMBH |
发明人 |
PFRENGLE, WALDEMAR;FRANK, MARKUS;KLEIN, THOMAS |
分类号 |
C07D473/06;A61K31/522 |
主分类号 |
C07D473/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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