发明名称 BENZAZEPINE COMPOUND
摘要 Provided is a compound which is useful as an agent for treating or preventing 5-HT2C receptor-related diseases, particularly incontinence such as stress urinary incontinence, urge urinary incontinence, mixed urinary incontinence, and the like, sexual dysfunction such as erectile dysfunction syndrome and the like, obesity, and the like. The present inventors have investigated compounds having a 5-HT2C receptor agonist activity and have found that the benzazepine compounds of the present invention have an excellent 5-HT2C receptor agonist activity, thereby completing the present invention. That is, the benzazepine compounds of the present invention have a 5-HT2C receptor agonist activity and can be used as an agent for treating or preventing 5-HT2C receptor-related diseases, particularly incontinence such as stress urinary incontinence, urge urinary incontinence, mixed urinary incontinence, and the like, sexual dysfunction such as erectile dysfunction syndrome and the like, obesity, and the like.
申请公布号 US2013012496(A1) 申请公布日期 2013.01.10
申请号 US201113583410 申请日期 2011.03.11
申请人 ASTELLAS PHARMA INC.;KOSHIO HIROYUKI;ASAI NORIO;TAKAHASHI TAISUKE;SHIMIZU TAKAFUMI;NAGAI YASUHITO;KAWABATA KEIKO;THOR KARL BRUCE 发明人 KOSHIO HIROYUKI;ASAI NORIO;TAKAHASHI TAISUKE;SHIMIZU TAKAFUMI;NAGAI YASUHITO;KAWABATA KEIKO;THOR KARL BRUCE
分类号 A61K31/55;A61P13/10;C07D487/04;C07D498/04 主分类号 A61K31/55
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