发明名称 OXAZETIDINE DERIVATIVES, PROCESS FOR PREPARING THEM AND USE THEREOF IN HUMAN MEDICINE AND IN COSMETICS
摘要 The present invention relates to the pharmaceutical field and in particular to the treatment of hypopigmentary pathologies and photosensitive dermatoses. More specifically, the invention relates to compounds that are agonists of the MC1R receptor and which exhibit reduced toxicity relative to the other compounds of the same class. These compounds have the general formula (I) below: in which: R1 represents a cyclopropylmethyl or a 4-hydroxybutyl group; R2 represents a hydrogen atom or a methyl group; and also the salts and enantiomers of the corresponding compounds of general formula (I).
申请公布号 CA2840606(A1) 申请公布日期 2013.01.03
申请号 CA20122840606 申请日期 2012.06.28
申请人 GALDERMA RESEARCH & DEVELOPMENT 发明人 BOUIX-PETER, CLAIRE
分类号 C07D403/12;A61K8/49;A61K31/4178;A61P17/00;A61Q5/02;A61Q19/00;A61Q19/10 主分类号 C07D403/12
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