发明名称 |
BICYCLIC RING SYSTEM SUBSTITUTED AMIDE FUNCTIONALISED PHENOLS AS MEDICAMENTS |
摘要 |
This invention relates to bicyclic ring system substituted amide functionalized phenols of general formula 1, their use as inhibitors of CXCR2 activity, pharmaceutical compositions containing the same, and methods of using the same as agents for treatment and/or prevention of respiratory or gastrointestinal complaints or diseases, inflammatory diseases of the joints, skin, or eyes, diseases of the peripheral or central nervous system or cancers, as well as pharmaceutical compositions which contain these compounds. |
申请公布号 |
US2012329773(A1) |
申请公布日期 |
2012.12.27 |
申请号 |
US201113324245 |
申请日期 |
2011.12.13 |
申请人 |
GIOVANNINI RICCARDO;HAMPRECHT DIETER;KISTLER BARBARA;LINGARD IAIN;BOEHRINGER INGELHEIM INTERNATIONAL GMBH |
发明人 |
GIOVANNINI RICCARDO;HAMPRECHT DIETER;KISTLER BARBARA;LINGARD IAIN |
分类号 |
A61K31/438;A61K31/397;A61K31/407;A61K31/437;A61K31/4985;A61K31/5383;A61K31/5386;A61K31/547;A61P1/00;A61P7/10;A61P11/00;A61P11/02;A61P11/06;A61P17/00;A61P19/02;A61P25/00;A61P27/02;A61P29/00;A61P31/00;A61P35/00;A61P37/08;C07D221/20;C07D471/04;C07D471/10;C07D487/04;C07D491/107;C07D498/04;C07D498/14;C07D498/20;C07D513/04;C07D513/10 |
主分类号 |
A61K31/438 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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