发明名称 STAT3/5 ACTIVATION INHIBITOR
摘要 The present invention provides a STAT3/5 activation inhibitor containing an aromatic compound represented by the general formula or a salt thereof as an active ingredient: Wherein X1 represents a nitrogen atom or a group —CH═, R1 represents a group —Z—R6, in which Z represents a group —CO—, a group —CH(OH)— or the like, R6 represents a 5- to 15-membered monocyclic, dicyclic or tricyclic saturated or unsaturated heterocyclic group having 1 to 4 nitrogen atoms, oxygen atoms or sulfur atoms, R2 represents a hydrogen atom or a halogen atom, Y represents a group —O—, a group —CO—, a group —CH(OH)— or a lower alkylene group, and A represents a group
申请公布号 US2012322807(A1) 申请公布日期 2012.12.20
申请号 US201213526283 申请日期 2012.06.18
申请人 SEKIGUCHI KAZUO;SUZUKI TAKASHI;OHBUCHI YUTAKA;OKUNO MITSUHIRO;OHI NAOTO;OHNISHI KENJI;MOTOYAMA MASAAKI;YOSHIDA KENJI;KODAMA TAKESHI;SUGIYAMA KAZUHISA;AKAMATSU SEIJI;KIYONO KUNIHIKO;YANAGIHARA YASUO;WATANABE TAKASHI;HAYASHI KAZUHIKO;TANAKA HIDEO;SUMIDA TAKUMI;OTSUKA PHARMACEUTICAL CO., LTD. 发明人 SEKIGUCHI KAZUO;SUZUKI TAKASHI;OHBUCHI YUTAKA;OKUNO MITSUHIRO;OHI NAOTO;OHNISHI KENJI;MOTOYAMA MASAAKI;YOSHIDA KENJI;KODAMA TAKESHI;SUGIYAMA KAZUHISA;AKAMATSU SEIJI;KIYONO KUNIHIKO;YANAGIHARA YASUO;WATANABE TAKASHI;HAYASHI KAZUHIKO;TANAKA HIDEO;SUMIDA TAKUMI
分类号 A61K31/496;A61P37/08 主分类号 A61K31/496
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