PROCESS FOR THE PREPARATION OF CRYSTALLINE FORMS OF AGOMELATINE AND NOVEL POLYMORPH THEREOF
摘要
The invention concerns a new process for the preparation of two crystalline forms of agomelatine, in particular a process for preparation of form I and a new form of agomelatine, here called form VII.
申请公布号
WO2012172387(A1)
申请公布日期
2012.12.20
申请号
WO2011IB03176
申请日期
2011.12.29
申请人
LABORATORIO CHIMICO INTERNAZIONALE S.P.A.;DE ANGELIS, BRUNO;GARIS, FARIS;DE GENNARO, SALVATORE;BERTOLINI, GIORGIO
发明人
DE ANGELIS, BRUNO;GARIS, FARIS;DE GENNARO, SALVATORE;BERTOLINI, GIORGIO