发明名称 |
PYRAZOLOPYRIDINE, PYRAZOLOPYRAZINE, PYRAZOLOPYRIMIDINE, PYRAZOLOTHIOPHENE AND PYRAZOLOTHIAZOLE COMPOUNDS AS MGLUR4 ALLOSTERIC POTENTIATORS, COMPOUNDS, AND METHODS OF TREATING NEUROLOGICAL DYSFUNCTION |
摘要 |
Pyrazolopyridine, pyrazolopyrazine, pyrazolopyrimidine, pyrazolothiophene and pyrazolothiazole compounds which are useful as allosteric potentiators/positive allosteric modulators of the metabotropic glutamate receptor subtype 4 (mGluR4); synthetic methods for making the compounds; pharmaceutical compositions comprising the compounds; and methods of using the compounds, for example, in treating neurological and psychiatric disorders or other disease state associated with glutamate dysfunction. |
申请公布号 |
EP2533639(A1) |
申请公布日期 |
2012.12.19 |
申请号 |
EP20110742910 |
申请日期 |
2011.02.11 |
申请人 |
VANDERBILT UNIVERSITY |
发明人 |
CONN, P., JEFFREY;LINDSLEY, CRAIG, W.;HOPKINS, COREY, R.;NISWENDER, COLLEEN, M.;GOGLIOTTI, ROCCO, D.;SALOVICH, JAMES, M.;ENGERS, DARREN, W.;CHEUNG, YIU-YIN |
分类号 |
A01N43/56;A61K31/415 |
主分类号 |
A01N43/56 |
代理机构 |
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代理人 |
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地址 |
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