发明名称 SUBSTITUTED PIPERIDINES AS GPR119 MODULATORS FOR THE TREATMENT OF METABOLIC DISORDERS
摘要 The present invention relates to compounds of general formula (I), wherein R1, Lp, HetAr, Ar, and n are as defined in the application, which have valuable pharmacological properties, and in particular bind to the GPR119 receptor and modulate its activity.
申请公布号 WO2012168315(A1) 申请公布日期 2012.12.13
申请号 WO2012EP60729 申请日期 2012.06.06
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH;NEUROCRINE BIOSCIENCES, INC.;HECKEL, ARMIN;HIMMELSBACH, FRANK;LANGKOPF, ELKE;NOSSE, BERND;ASHWEEK, NEIL, J.;HARRIOTT, NICOLE 发明人 HECKEL, ARMIN;HIMMELSBACH, FRANK;LANGKOPF, ELKE;NOSSE, BERND;ASHWEEK, NEIL, J.;HARRIOTT, NICOLE
分类号 C07D413/14;A61K31/454;A61K31/4545;A61K31/497;A61K31/506;A61P3/10;C07D401/14 主分类号 C07D413/14
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