发明名称 |
SUBSTITUTED INDOLYL ALKYL AMINO DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE |
摘要 |
<p>THIS INVENTION COMPRISES THE NOVEL COMPOUNDS OF FORMULA (?) WHEREIN R¹, R², R³, X AND Y HAVE DEFINED MEANINGS, HAVING HISTONE DEACETYLASE INHIBITING ENZYMATIC ACTIVITY, THEIR PREPARATION, COMPOSITIONS CONTAINING THEM AND THEIR USE AS A MEDICINE.</p> |
申请公布号 |
MY147316(A) |
申请公布日期 |
2012.11.30 |
申请号 |
MY2005PI03453 |
申请日期 |
2005.07.27 |
申请人 |
JANSSEN PHARMACEUTICA N.V. |
发明人 |
MARC GUSTAAF CELINE VERDONCK;PATRICK RENE ANGIBAUD;BRUNO ROUX;ISABELLE NOELLE CONSTANCE PILATTE;PETER TEN HOLTE;JANINE ARTS;KRISTOF VAN EMELEN |
分类号 |
C07D401/14;A61K31/506;C07D405/14;C07D409/14 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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