发明名称 |
1,3,4-OXADIAZOLE-2-CARBOXAMIDE COMPOUND |
摘要 |
Provided is a 1,3,4-oxadiazole-2-carboxamide compound which has STAT3 inhibitory activity and is useful as an anticancer agent. Provided is a 1,3,4-oxadiazole-2-carboxamide compound represented by formula (I) or a pharmacologically acceptable salt thereof (in the formula, Ar represents a furyl group or the like; R1 represents a hydrogen atom or the like; and —X—Y represents a diaryl group such as a biphenyl group).
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申请公布号 |
US2012302524(A1) |
申请公布日期 |
2012.11.29 |
申请号 |
US201013519707 |
申请日期 |
2010.12.28 |
申请人 |
ASAI AKIRA;MATSUNO KENJI;OGO NAOHISA;TAKAHASHI OSAMU;MASUDA YOSHIAKI;MUROYA AYUMU;AKIYAMA YASUTO;ASHIZAWA TADASHI;OKAWARA TADASHI;GENERAL INCORPORATED ASSOCIATION PHARMA VALLEY PROJECT SUPPORTING ORGANIZATION;PHARMA DESIGN, INC.;KABUSHIKI KAISHA YAKULT HONSHA;KUMAMOTO HEALTH SCIENCE UNIVERSITY;SHIZUOKA PREFECTURE |
发明人 |
ASAI AKIRA;MATSUNO KENJI;OGO NAOHISA;TAKAHASHI OSAMU;MASUDA YOSHIAKI;MUROYA AYUMU;AKIYAMA YASUTO;ASHIZAWA TADASHI;OKAWARA TADASHI |
分类号 |
A61K31/4245;A61K31/437;A61K31/4439;A61K31/454;A61K31/4545;A61K31/4709;A61K31/496;A61K31/498;A61K31/5377;A61K31/541;A61K31/55;A61K31/695;A61P35/00;C07D413/04;C07D413/14;C07D487/04;C07D513/04;C07F7/10 |
主分类号 |
A61K31/4245 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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