发明名称 PHENYL-THIAZOLYL INHIBITORS OF PRO-MATRIX METALLOPROTEINASE ACTIVATION
摘要 This invention relates to phenyl thiazole I and its therapeutic and prophylactic uses, wherein the variables Rz, Q, J, R1, R3, R5, R6, and R7 are defined in the specification. Disorders treated and/or prevented include rheumatoid arthritis.
申请公布号 US2012302569(A1) 申请公布日期 2012.11.29
申请号 US201213479395 申请日期 2012.05.24
申请人 JACKSON PAUL FRANCIS;LEONARD KRISTI ANNE;BARBAY JOSEPH KENT;WANG AIHUA;TOUNGE BRETT ANDREW;ZHANG YAN;MAHAROOF UMAR S.M. 发明人 JACKSON PAUL FRANCIS;LEONARD KRISTI ANNE;BARBAY JOSEPH KENT;WANG AIHUA;TOUNGE BRETT ANDREW;ZHANG YAN;MAHAROOF UMAR S.M.
分类号 A61K31/427;A61K31/4439;A61K31/444;A61K31/454;A61K31/496;A61K31/5377;A61P1/00;A61P1/02;A61P1/04;A61P1/16;A61P9/00;A61P9/10;A61P9/12;A61P11/00;A61P11/06;A61P13/12;A61P17/02;A61P19/02;A61P25/00;A61P25/06;A61P29/00;A61P35/00;C07D417/10;C07D417/12;C07D417/14 主分类号 A61K31/427
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