PROCESS FOR THE PREPARATION OF a-SUBSTITUTED KETONES AND THEIR APPLICATION IN SYNTHESIS OF PHARMACEUTICALLY ACTIVE COMPOUNDS
摘要
The present invention relates to a novel one step preparation of 6-methoxy-2-phenyl-tetralone starting from 6-methoxy-tetralone and its use as an intermediate in the synthesis of pharmaceutically active compounds.
申请公布号
WO2012159981(A2)
申请公布日期
2012.11.29
申请号
WO2012EP59236
申请日期
2012.05.18
申请人
LEK PHARMACEUTICALS D.D.;GAZIC SMILOVIC, IVANA;SEECHURN, CARIN;COLACOT, THOMAS J.
发明人
GAZIC SMILOVIC, IVANA;SEECHURN, CARIN;COLACOT, THOMAS J.