发明名称 DERIVATIVES OF PYRIMIDO [6,1-A] ISOQUINOLIN-4-ONE
摘要 The present invention relates to derivatives of pyrimido[6,1-a]isoquinolin-4-one and their application as inhibitors of phosphodiesterase (PDE) isoenzymes. More particularly the invention relates to derivatives of pyrimido[6,1-a]isoquinolin-4-one and their use in medicine for example as bronchodilators with anti-inflammatory properties.
申请公布号 US2012302533(A1) 申请公布日期 2012.11.29
申请号 US201213568754 申请日期 2012.08.07
申请人 OXFORD ALEXANDER WILLIAM;JACK DAVID;VERONA PHARMA PLC 发明人 OXFORD ALEXANDER WILLIAM;JACK DAVID
分类号 A61K31/519;A61K9/12;A61K31/56;A61P11/00;A61P11/06;A61P11/08;A61P29/00;A61P43/00;C07D471/04 主分类号 A61K31/519
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