发明名称 3-POLYLYSINE CONJUGATES AND THE USE THEREOF
摘要 Conjugate comprises at least one carboxyl group-containing compound and an oligomer, where the oligomer: comprises peptidically crosslinked monomer units; is formed from more than 50%, relative to the number of monomer units, of epsilon -lysine monomer units; or comprises at least 10 consecutive monomer units that are formed from at least up to 70%, relative to the number of monomer units, of epsilon -lysine monomer units. Independent claims are included for: (1) the preparation of the conjugate comprising providing the oligomers, as above per se, and conjugating at least one optionally activated carboxylic group-containing compound to the oligomer; and (2) a kit, for preparing pharmaceutical composition (preferably a therapeutic or image enhancing composition), comprising the above conjugate.
申请公布号 ZA201201218(B) 申请公布日期 2012.11.28
申请号 ZA20120001218 申请日期 2012.02.17
申请人 MERCK PATENT GMBH 发明人 KUEBELBECK ARMIN;MIER WALTER;HABERKORN UWE;LARBIG GREGOR;BEIJER BARBRO
分类号 A61K 主分类号 A61K
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