摘要 |
<p>A heterocyclic compound represented by general formula (I)
[wherein R 1 represents an optionally protected amino group, or an optionally substituted C 1-6 alkyl group; R 2 and R 3 independently represent a C 1-2 alkyl group; X represents a hydrogen atom, or a halogen atom; Z 1 represents C-R 4 (wherein R 4 represents a hydrogen atom, a halogen atom, an optionally protected amino group, or a C 1-6 alkylsulfonyl group), or N; Z 2 represents C-R 5 (wherein, R 5 represents a hydrogen atom, a hydrogen atom, a halogen atom, an optionally protected amino group, or a C 1-6 alkylsulfonyl group), or N; Z 3 represents C-R 6 (wherein R 6 represents a hydrogen atom, a hydrogen atom, a halogen atom, an optionally protected amino group, or a C 1-6 alkylsulfonyl group ), or N; Z 4 represents C-R 7 (wherein, R 7 represents a hydrogen atom, a hydrogen atom, a halogen atom, an optionally protected amino group, or a C 1-6 alkylsulfonyl group), or N; Z represents CH or N; and A represents a methylene group, or a bond] or a salt thereof, which has an excellent anti-HIV activity and is thereof useful as an anti-HIV agent.</p> |
申请人 |
TOYAMA CHEMICAL CO., LTD. |
发明人 |
OONISHI, YUJI;AWASAGUCHI, KENICHIRO;NOMURA, NOBUHIKO;TOHDO, KEISUKE;KAWAI, HYOUEI;WAKATSUKI, TOMOMI |