发明名称 NOVEL CRYSTALLINE SALTS OF ASENAPINE
摘要 The present invention relates to novel crystalline salts of Asenapine and to methods of their preparation. In particular, the invention relates to crystalline Asenapine salts of tartaric acid or succinic acid, wherein the salts are e.g. selected from the group consisting of Asenapine D, L-tartrate hydrate form A, Asenapine D, L-tartrate hydrate form B, Asenapine D, L-tartrate anhydrous form, Asenapine succinate form X, Asenapine succinate form, and Asenapine succinate form II. Furthermore the present invention relates to pharmaceutical compositions comprising the novel salts and to the novel salts for use in the treatment of psychotic diseases or disorders.
申请公布号 WO2012156384(A1) 申请公布日期 2012.11.22
申请号 WO2012EP58964 申请日期 2012.05.15
申请人 SANDOZ AG;BLATTER, FRITZ;REICHENBAECHER, KATHARINA 发明人 BLATTER, FRITZ;REICHENBAECHER, KATHARINA
分类号 C07D491/044;A61K31/407;A61P25/18 主分类号 C07D491/044
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