发明名称 |
NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS |
摘要 |
<p>Provided herein are novel and selective high affinityα3β4 nicotinic acetycholine receptor ligands and pharmaceutical compositions thereof. In other embodiments, provided herein are methods of treatment, prevention, or amelioration of a variety of medical disorders such as, for example, drug addiction or pain using the compounds and compositions disclosed herein. In still other embodiments, provided herein are methods of selectively antagonizing receptors such as, for example, theα3β4 nicotinic acetycholine receptor using the compounds and compositions disclosed herein.</p> |
申请公布号 |
EP2523562(A1) |
申请公布日期 |
2012.11.21 |
申请号 |
EP20110732326 |
申请日期 |
2011.01.11 |
申请人 |
ASTRAEA THERAPEUTICS, LLC |
发明人 |
ZAVERI, NURULAIN, T.;JIANG, FAMING;TOLL, LAWRENCE |
分类号 |
A61K31/439;A61P25/30;C07D451/14 |
主分类号 |
A61K31/439 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|