发明名称 |
METHOD FOR PREPARING TETRAZOLE METHANESULFONIC ACID SALTS, AND NOVEL COMPOUND USED IN SAME |
摘要 |
<p>According to the present invention, a method for preparing tetrazole methanesulfonic acid salts comprises an acylation reaction using a novel 4-iodine-4H-chromene-2-carbothionic acid S-benzothiazole-2-yl ester. The method of the present invention can shorten a reaction time and improve safety as compared to conventional methods, and can prepare high-purity tetrazole methanesulfonic acid salts at a high yield rate without using a column chromatography method.</p> |
申请公布号 |
EP2524916(A2) |
申请公布日期 |
2012.11.21 |
申请号 |
EP20110733103 |
申请日期 |
2011.01.14 |
申请人 |
HANMI SCIENCE CO., LTD. |
发明人 |
BANG, KEUK CHAN;PARK, BUM WOO;CHOI, JONG WON;LEE, JAE CHUL;AN, YONG HOON;AHN, YOUNG GIL;KIM, MAENG SUP |
分类号 |
C07D405/14;C07D403/02;C07D403/10;C07D405/12;C07D417/12 |
主分类号 |
C07D405/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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