发明名称 INDAZOLYL ESTER AND AMIDE DERIVATIVE FOR TREATMENT OF GLUCOCORTICOID RECEPTOR-MEDIATED DISORDER
摘要 <P>PROBLEM TO BE SOLVED: To provide novel indazolyl ester or amide derivatives, pharmaceutical compositions comprising such derivatives, processes for preparing such novel derivatives, and the use of such derivatives as medicaments, which are suitable for the treatment of an inflammatory disease state. <P>SOLUTION: This invention relates to: compounds of formula (I); pharmaceutical compositions comprising such derivatives; processes for preparing such novel derivatives; and the use of such derivatives as medicaments. <P>COPYRIGHT: (C)2013,JPO&INPIT
申请公布号 JP2012224647(A) 申请公布日期 2012.11.15
申请号 JP20120184346 申请日期 2012.08.23
申请人 ASTRAZENECA AB;BAYER PHARMA AG 发明人 BERGER MARKUS;DAHMEN JAN;ERIKSSON ANDERS;GABOS BALINT;HANSSON THOMAS;HEMMERLING MARTIN;HENRIKSSON KRISTER;IVANOVA SVETLANA;MATTI LEPISTOE;MCKERRECHER DARREN;MAGNUS MUNCK AF ROSENSCHOELD;NILSSON STINABRITT;REHWINKEL HARTMUT;TAFLIN CAMILLA;EDMAN KARL
分类号 C07D231/56;A61K31/416;A61K31/4178;A61K31/4184;A61K31/4192;A61K31/4196;A61K31/422;A61K31/4245;A61K31/427;A61K31/428;A61K31/437;A61K31/4439;A61K31/4709;A61K31/501;A61K31/506;A61K31/5377;A61K45/00;A61P1/00;A61P1/16;A61P3/04;A61P3/10;A61P5/00;A61P5/16;A61P7/00;A61P7/06;A61P9/00;A61P9/06;A61P9/10;A61P9/12;A61P11/00;A61P11/02;A61P11/06;A61P11/08;A61P13/12;A61P17/00;A61P17/04;A61P17/06;A61P17/14;A61P19/02;A61P19/10;A61P21/00;A61P25/00;A61P25/22;A61P25/24;A61P25/28;A61P27/02;A61P29/00;A61P35/00;A61P35/02;A61P35/04;A61P37/06;A61P37/08;A61P43/00;C07D401/04;C07D401/12;C07D403/04;C07D403/12;C07D405/12;C07D405/14;C07D409/12;C07D413/12;C07D417/12;C07D417/14;C07D471/04 主分类号 C07D231/56
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