发明名称 |
3,4,4A,10B-TETRAHYDRO-1H-THIOPYRANO-[4,3-c] ISOQUINOLINE DERIVATIVES |
摘要 |
The compounds of Formula (1), in which A, R1, R2, R3 and R5 have the meanings as given in the description, are novel effective inhibitors of type 4 and 5 phosphodiesterase. |
申请公布号 |
US2012289474(A1) |
申请公布日期 |
2012.11.15 |
申请号 |
US201013515214 |
申请日期 |
2010.12.15 |
申请人 |
FLOCKERZI DIETER;STENGEL THOMAS;MANN ALEXANDER;OHMER HARALD;KAUTZ ULRICH;WEINBRENNER STEFFEN;FISCHER STEFAN;ZITT CHRISTOF;HATZELMANN ARMIN;DUNKERN TORSTEN;HESSLINGER CHRISTIAN;MAIER THOMAS;TENOR HERMANN;BRAUN CLEMENS;KUELZER RAIMUND;MARX DEGENHARD;NYCOMED GMBH |
发明人 |
FLOCKERZI DIETER;STENGEL THOMAS;MANN ALEXANDER;OHMER HARALD;KAUTZ ULRICH;WEINBRENNER STEFFEN;FISCHER STEFAN;ZITT CHRISTOF;HATZELMANN ARMIN;DUNKERN TORSTEN;HESSLINGER CHRISTIAN;MAIER THOMAS;TENOR HERMANN;BRAUN CLEMENS;KUELZER RAIMUND;MARX DEGENHARD |
分类号 |
A61K31/519;A61K31/5585;A61K31/56;A61K31/59;A61K31/7048;A61P7/02;A61P7/10;A61P9/12;A61P11/00;A61P11/06;A61P11/08;A61P31/00;A61P37/06;C07D495/04 |
主分类号 |
A61K31/519 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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