发明名称 3,4,4A,10B-TETRAHYDRO-1H-THIOPYRANO-[4,3-c] ISOQUINOLINE DERIVATIVES
摘要 The compounds of Formula (1), in which A, R1, R2, R3 and R5 have the meanings as given in the description, are novel effective inhibitors of type 4 and 5 phosphodiesterase.
申请公布号 US2012289474(A1) 申请公布日期 2012.11.15
申请号 US201013515214 申请日期 2010.12.15
申请人 FLOCKERZI DIETER;STENGEL THOMAS;MANN ALEXANDER;OHMER HARALD;KAUTZ ULRICH;WEINBRENNER STEFFEN;FISCHER STEFAN;ZITT CHRISTOF;HATZELMANN ARMIN;DUNKERN TORSTEN;HESSLINGER CHRISTIAN;MAIER THOMAS;TENOR HERMANN;BRAUN CLEMENS;KUELZER RAIMUND;MARX DEGENHARD;NYCOMED GMBH 发明人 FLOCKERZI DIETER;STENGEL THOMAS;MANN ALEXANDER;OHMER HARALD;KAUTZ ULRICH;WEINBRENNER STEFFEN;FISCHER STEFAN;ZITT CHRISTOF;HATZELMANN ARMIN;DUNKERN TORSTEN;HESSLINGER CHRISTIAN;MAIER THOMAS;TENOR HERMANN;BRAUN CLEMENS;KUELZER RAIMUND;MARX DEGENHARD
分类号 A61K31/519;A61K31/5585;A61K31/56;A61K31/59;A61K31/7048;A61P7/02;A61P7/10;A61P9/12;A61P11/00;A61P11/06;A61P11/08;A61P31/00;A61P37/06;C07D495/04 主分类号 A61K31/519
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