发明名称 |
S-TRIAZOLYL ALPHA-MERCAPTO ACETANILIDES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE |
摘要 |
A series of S-triazolyl α-mercaptoacetanilides having general structure (1) are provided, where Q is CO2H, CONR2, SO3H, or SO2NR2. The compounds inhibit several variants of the reverse transcriptase of HIV, and are useful in the treatment of HIV infections. |
申请公布号 |
US2012283301(A1) |
申请公布日期 |
2012.11.08 |
申请号 |
US201213552443 |
申请日期 |
2012.07.18 |
申请人 |
GIRARDET JEAN-LUC;KOH YUNG-HYO;DE LA ROSA MARTHA;GUNIC ESMIR;HONG ZHI;LANG STANLEY;KIM WOO-HONG;ARDEA BIOSCIENCES INC. |
发明人 |
GIRARDET JEAN-LUC;KOH YUNG-HYO;DE LA ROSA MARTHA;GUNIC ESMIR;HONG ZHI;LANG STANLEY;KIM WOO-HONG |
分类号 |
A61K31/4196;A61P31/18;C07D249/12 |
主分类号 |
A61K31/4196 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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