发明名称 S-TRIAZOLYL ALPHA-MERCAPTO ACETANILIDES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE
摘要 A series of S-triazolyl α-mercaptoacetanilides having general structure (1) are provided, where Q is CO2H, CONR2, SO3H, or SO2NR2. The compounds inhibit several variants of the reverse transcriptase of HIV, and are useful in the treatment of HIV infections.
申请公布号 US2012283301(A1) 申请公布日期 2012.11.08
申请号 US201213552443 申请日期 2012.07.18
申请人 GIRARDET JEAN-LUC;KOH YUNG-HYO;DE LA ROSA MARTHA;GUNIC ESMIR;HONG ZHI;LANG STANLEY;KIM WOO-HONG;ARDEA BIOSCIENCES INC. 发明人 GIRARDET JEAN-LUC;KOH YUNG-HYO;DE LA ROSA MARTHA;GUNIC ESMIR;HONG ZHI;LANG STANLEY;KIM WOO-HONG
分类号 A61K31/4196;A61P31/18;C07D249/12 主分类号 A61K31/4196
代理机构 代理人
主权项
地址