Disclosed is asenapine phosphate of formula (I) and its enantiomer (I) which can be used to prepare asenapine maleate. Further disclosed is a monoclinic crystalline form of asenapine maleate.
申请公布号
WO2012150538(A1)
申请公布日期
2012.11.08
申请号
WO2012IB52151
申请日期
2012.04.30
申请人
OLON SPA;FRIGOLI, SAMUELE;LONGONI, DAVIDE;DANELLI, TAMARA;ALPEGIANI, MARCO
发明人
FRIGOLI, SAMUELE;LONGONI, DAVIDE;DANELLI, TAMARA;ALPEGIANI, MARCO