发明名称 |
CRYSTAL OF HYPOXIA INDUCIBLE FACTOR 1 ALPHA PROLYL HYDROXYLASE |
摘要 |
The crystal structure of ligand-bound EGLN1 catalytic domain of prolyl hydroxylase is disclosed. These coordinates are useful in computer aided drug design for identifying compounds that regulate EGLN1 prolyl hydroxylase and thereby regulate HIF-regulated disorders. |
申请公布号 |
US2012282627(A1) |
申请公布日期 |
2012.11.08 |
申请号 |
US201113230548 |
申请日期 |
2011.09.12 |
申请人 |
EVDOKIMOV ARTEM GENNADY;KAWAMOTO RICHARD MASARU;BOYER ANGELIQUE SUN;MEKEL MARLENE JAN;POKROSS MATTHEW EUGENE;WALTER, JR. RICHARD LEE |
发明人 |
EVDOKIMOV ARTEM GENNADY;KAWAMOTO RICHARD MASARU;BOYER ANGELIQUE SUN;MEKEL MARLENE JAN;POKROSS MATTHEW EUGENE;WALTER, JR. RICHARD LEE |
分类号 |
G01N33/573;C12Q1/34;G06F19/10 |
主分类号 |
G01N33/573 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|