发明名称
摘要 The present invention relates to the Janus kinase (JAK) inhibitors 3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]octanenitrile or 3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]heptanenitrile, as well as its compositions and methods of use, which is useful in the treatment of JAK-associated diseases including, for example, inflammatory and autoimmune disorders, skin disorders, cancer, and other diseases.
申请公布号 JP2012527481(A) 申请公布日期 2012.11.08
申请号 JP20120512056 申请日期 2010.05.21
申请人 发明人
分类号 C07D487/04;A61K9/06;A61K9/08;A61K9/107;A61K9/70;A61K31/519;A61P1/00;A61P1/04;A61P3/10;A61P9/10;A61P13/12;A61P17/00;A61P17/06;A61P19/02;A61P21/04;A61P25/00;A61P27/02;A61P29/00;A61P31/12;A61P31/14;A61P31/18;A61P31/20;A61P35/02;A61P37/00;A61P37/06;A61P37/08;A61P43/00 主分类号 C07D487/04
代理机构 代理人
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