发明名称 |
Propofol analogs, process for their preparation, and methods of use |
摘要 |
<p>The invention provides para substituted dialkylphenol derivatives of propofol. The invention further provides pharmaceutical compositions comprising such analogs, methods for preparing such analogs, and methods of using such analogs to induce general anesthesia, sedation, and/or hypnotic or sleep effects in a patient.</p> |
申请公布号 |
EP2520290(A1) |
申请公布日期 |
2012.11.07 |
申请号 |
EP20110009745 |
申请日期 |
2004.12.23 |
申请人 |
ABRAXIS BIOSCIENCE, LLC |
发明人 |
TAO, CHUNLIN;YU, CHENGZHI;DESAI, NEIL P.;TRIEU, VUONG |
分类号 |
A61K31/275;A61K31/05;A61K31/095;A61K31/12;A61K31/15;A61P23/00;A61P25/20;C07C39/367;C07C39/373;C07C45/00;C07C45/46;C07C49/83;C07C49/84;C07C69/78;C07C205/45;C07C225/22;C07C235/84;C07C251/48;C07C255/56;C07C309/87;C07C311/29;C07C317/24;C07C325/02;C07D317/54;C07D317/56;C07D317/58 |
主分类号 |
A61K31/275 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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