发明名称 AN IMPROVED PROCESS FOR THE PREPARATION OF SILODOSIN
摘要 <p>The present invention provides a process for the preparation of Silodosin of Formula (I). More particularly, the present invention provides the process for preparation of tartrate salt of 3-[7-cyano-5[(2R)-2-({2-[2-(2,2,2- trifluoroethoxy)phenoxy]ethyl}amino)propyl]-2, 3-dihydro-1H-indol-1 -yl }propyl benzoate of Formula (IV), which is a precursor in the preparation of Silodosin.</p>
申请公布号 WO2012147019(A1) 申请公布日期 2012.11.01
申请号 WO2012IB52015 申请日期 2012.04.21
申请人 ORCHID CHEMICALS AND PHARAMCEUTICALS LIMITED;REGURI, BUCHI, REDDY;THIRUMANI, VENKATESHWAR, GOUD;NAGABUSHANAM, NAGAMANI;RAMASAMY, KAMALA;DEVINENI, SURESH;SHAIK, MAHABOOB, BASHA 发明人 REGURI, BUCHI, REDDY;THIRUMANI, VENKATESHWAR, GOUD;NAGABUSHANAM, NAGAMANI;RAMASAMY, KAMALA;DEVINENI, SURESH;SHAIK, MAHABOOB, BASHA
分类号 C07D209/08 主分类号 C07D209/08
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