发明名称 |
PRODRUGS OF COMPOUNDS THAT INHIBIT TRPV1 RECEPTOR |
摘要 |
Compounds of formula (I) wherein A, R1, R2, and R3 are defined in the specification, and which are useful as therapeutic compounds particularly for treating disorders or conditions associated with inflammation, pain, bladder overactivity, urinary incontinence, and other disorders caused by or exacerbated by TRPV1. |
申请公布号 |
US2012277190(A1) |
申请公布日期 |
2012.11.01 |
申请号 |
US201213544130 |
申请日期 |
2012.07.09 |
申请人 |
GOMTSYAN ARTHUR R.;BAYBURT EROL K.;KOENIG JOHN R.;MARSH KENNAN C.;SCHMIDT, JR. ROBERT G.;LEE CHIH-HUNG;WANG WEILI;DAANEN JEROME F.;BROWN BRIAN S. |
发明人 |
GOMTSYAN ARTHUR R.;BAYBURT EROL K.;KOENIG JOHN R.;MARSH KENNAN C.;SCHMIDT, JR. ROBERT G.;LEE CHIH-HUNG;WANG WEILI;DAANEN JEROME F.;BROWN BRIAN S. |
分类号 |
A61K31/5377;A61K31/416;A61K31/454;A61K31/675;A61P13/10;A61P25/00;C07D231/56;C07D401/12;C07D413/06;C07F9/09 |
主分类号 |
A61K31/5377 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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