发明名称 |
RADIOIODINATED TROPANE DERIVATIVES |
摘要 |
The present invention provides novel radio iodinated tropanes incorporating triazole or isoxazole rings. Also provided are methods of preparation of said tropanes from functionalised tropane precursors, using click cycloaddition chemistry, as well as radiopharmaceutical compositions comprising such radio iodinated tropanes. The invention also provides in vivo imaging methods using the radio iodinated tropanes. |
申请公布号 |
EP2516427(A1) |
申请公布日期 |
2012.10.31 |
申请号 |
EP20100799019 |
申请日期 |
2010.12.21 |
申请人 |
GE HEALTHCARE LIMITED |
发明人 |
AVORY, MICHELLE, EMMA;WADSWORTH, HARRY, JOHN;NAIRNE, JAMES DOMETT |
分类号 |
C07D451/02 |
主分类号 |
C07D451/02 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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