发明名称 Novel antifungal 5,6-dihydro-4-[(difluoroethyl)phenyl]-4H-pyrrolo[1,2-a][1,4]-benzodiazepine and 4-(diflouroethyl)phenyl-6H-pyrrolo[1,2-a][1,4]benzodiazepenine derivatives
摘要 <p>The present invention concerns novel compounds of Formula (I): wherein R1, R2, R3, R4, R5 and R6 have the meaning defined in the claims. The compounds according to the present invention are active mainly against dermatophytes and systemic fungal infections. The invention further relates to processes for preparing such novel compounds, pharmaceutical compositions comprising said compounds as an active ingredient as well as the use of said compounds as a medicament.</p>
申请公布号 AP201206502(D0) 申请公布日期 2012.10.31
申请号 AP20120006502 申请日期 2011.06.01
申请人 JANSSEN PHARMACEUTICA NV 发明人 WIT KELLY DE;MAES LOUISE JULES ROGER MARIE;MEERPOEL LIEVEN
分类号 C07D487/04;A61K31/5517;A61P31/10 主分类号 C07D487/04
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