发明名称 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONIST
摘要 A compound of the formula (I) wherein the variables X 1 to X 10 , R 1 to R 7 including R 3' , E, v, y, z, A and B are as described, or a pharmaceutically acceptable salt, solvate, enantiomer, racemate, diastereomer or mixtures thereof, useful for the treatment, prevention or amelioration of obesity and Related Diseases is disclosed.
申请公布号 PL212616(B1) 申请公布日期 2012.10.31
申请号 PL20030376057 申请日期 2003.09.17
申请人 ELI LILLY AND COMPANY 发明人 BLANCO-PILLADO MARIA-JESUS;CHAPPELL MARK DONALD;DE LA TORRE MARTA GARCIA;DIAZ BUEZO NURIA;FRITZ JAMES ERWIN;HOLLOWAY WILLIAM GLEN;MATT JAMES EDWARD JUNIOR;MITCH CHARLES HOWARD;PEDREGAL-TERCERO CONCEPCION;QUIMBY STEVEN JAMES;SIEGEL MILES GOODMAN;SMITH DANA RAE;STUCKY RUSSELL DEAN;TAKEUCHI KUMIKO;THOMAS ELIZABETH MARIE;WOLFE CHAD NOLAN
分类号 C07D241/24;A61K31/351;A61K31/4412;A61K31/4433;A61K31/497;A61P3/04;C07C43/20;C07C235/46;C07D213/38;C07D213/64;C07D213/643;C07D213/78;C07D213/81;C07D213/82;C07D217/04;C07D237/24;C07D307/14;C07D333/20;C07D401/06;C07D401/12;C07D401/14;C07D405/10;C07D405/12;C07D409/12;C07D409/14;C07D413/12;C07D417/12;C07D417/14 主分类号 C07D241/24
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