发明名称 BICYCLIC AMINE DERIVATIVES AS TYROSINE KINASE INHIBITORS
摘要 FIELD: chemistry. ^ SUBSTANCE: invention relates to novel bicyclic heterocyclic derivatives, which are compounds of formula where values of X1-X5, A, B, R1, R2, q are given in claim 1, as well as pharmaceutical compositions containing said compounds, and use of said compounds to treat cancer. ^ EFFECT: high efficiency of treatment. ^ 22 cl, 43 ex
申请公布号 RU2465275(C2) 申请公布日期 2012.10.27
申请号 RU20090128186 申请日期 2007.12.21
申请人 ASTEKS TERAP'JUTIKS LIMITED 发明人 BERDINI VALERIO;BEZONG GILBERT EHBAJ;KALLAGAN OUEHN;KARR MARIJA GRATSIJA;KONGRIV MAJLZ STJUART;DZHILL EHDRIAN LIEHM;GRIFFITS-DZHOUNZ SHARLOTT MEHRI;MEHDIN EHNDRJU;MJURREJ KRISTOFER UILL'JAM;NIDZHAR RADZHDIP KAUR;O'BRAJEN MAJKL ALISTEHR;PAJK EHNDRJU;SAKSTI GORDON;TEHJLOR RICHARD DEHVID;VIKERSTAFF EHMMA
分类号 A61K31/4375;A61P35/00;C07D471/04;C07D487/04 主分类号 A61K31/4375
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