发明名称 |
PROCESS FOR PREPARING SUBSTITUTED 1-O-ACYL-2-DEOXY-2-FLUORO-4-THIO-ß-D-ARABINOFURANOSES |
摘要 |
<p>The present invention relates to a process for preparing 1-O-acyl-2-deoxy-2-ftuoro-4-thio-²-D-arabinofuranoses having formula I and intermediates thereof:
wherein R 1 represents -C(O)-C 1 -C 6 -alkyl or -C(O)-aryl; and R 2 represents C 1 -C 6 -alkyl, C 1 -C 4 -perfluoroalkyl or aryl.</p> |
申请公布号 |
EP2513081(A1) |
申请公布日期 |
2012.10.24 |
申请号 |
EP20100801279 |
申请日期 |
2010.12.03 |
申请人 |
LIBRAMEDICINA, INC. |
发明人 |
VOIGTLANDER, DAVID;SANDER, MICHAEL;HARRE, MICHAEL |
分类号 |
C07D317/18;C07D333/32;C07D333/78 |
主分类号 |
C07D317/18 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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