发明名称 |
ENANTIOMERICALLY PURE AMINOHETEROARYL COMPOUNDS AS PROTEIN KINASE INHIBITORS |
摘要 |
Enantiomerically pure compound of formula 1 are provided, as well as methods for their synthesis and use. Preferred compounds are potent inhibitors of the c-Met protein kinase, and are useful in the treatment of abnormal cell growth disorders, such as cancers. |
申请公布号 |
US2012263706(A1) |
申请公布日期 |
2012.10.18 |
申请号 |
US201213537759 |
申请日期 |
2012.06.29 |
申请人 |
CUI JINGRONG JEAN;FUNK LEE ANDREW;JIA LEI;KUNG PEI-PEI;MENG JERRY JIALUN;NAMBU MITCHELL DAVID;PAIRISH MASON ALAN;SHEN HONG;TRAN-DUBE MICHELLE;AGOURON PHARMACEUTICALS, INC. |
发明人 |
CUI JINGRONG JEAN;FUNK LEE ANDREW;JIA LEI;KUNG PEI-PEI;MENG JERRY JIALUN;NAMBU MITCHELL DAVID;PAIRISH MASON ALAN;SHEN HONG;TRAN-DUBE MICHELLE |
分类号 |
A61K31/4418;A61K31/4439;A61K31/4545;A61K31/496;A61K31/4965;A61K31/497;A61K39/395;A61P35/00;A61P35/02;C07D213/73;C07D241/20;C07D401/04;C07D401/10;C07D401/14;C07D403/04;C07D403/10;C07D521/00 |
主分类号 |
A61K31/4418 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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