发明名称 SUBSTITUTED CYCLOPROPYL COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT
摘要 Substituted cyclopropyl compounds of the formula I: and pharmaceutically acceptable salts thereof are disclosed as useful for treating or preventing type 2 diabetes and similar conditions. The compounds are useful as agonists of the G-protein coupled receptor GPR-119. Pharmaceutical compositions and methods of treatment are also included
申请公布号 WO2012138845(A1) 申请公布日期 2012.10.11
申请号 WO2012US32303 申请日期 2012.04.05
申请人 MERCK SHARP & DOHME CORP.;EDMONDSON, SCOTT;GUO, ZHIQIANG;GEISS, WILLIAM, B.;WOOD, HAROLD, B.;STAMFORD, ANDREW, W.;MILLER, MICHAEL, W.;DEMONG, DUANE, E.;MORRIELLO, GREGORI, J.;ANAND, RAJAN;COLANDREA, VINCENT, J.;MACALA, MEGAN;MALETIC, MILANA;ZHU, CHENG;ZHU, YUPING;SUN, WANYING;ZHAO, KAKE;HUANG, YONG;HARRIS, JOEL, M.;CHANG, LEHUA;KAR, NAM FUNG;HU, ZHIYONG;WANG, LIPING;WANG, BOWEI;LIU, PING;SZEWCZYK, JASON, W. 发明人 EDMONDSON, SCOTT;GUO, ZHIQIANG;GEISS, WILLIAM, B.;WOOD, HAROLD, B.;STAMFORD, ANDREW, W.;MILLER, MICHAEL, W.;DEMONG, DUANE, E.;MORRIELLO, GREGORI, J.;ANAND, RAJAN;COLANDREA, VINCENT, J.;MACALA, MEGAN;MALETIC, MILANA;ZHU, CHENG;ZHU, YUPING;SUN, WANYING;ZHAO, KAKE;HUANG, YONG;HARRIS, JOEL, M.;CHANG, LEHUA;KAR, NAM FUNG;HU, ZHIYONG;WANG, LIPING;WANG, BOWEI;LIU, PING;SZEWCZYK, JASON, W.
分类号 A01N43/54;A01N43/40;A61K31/445;A61K31/505 主分类号 A01N43/54
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